Pycup—A Bifunctional, Cage-like Ligand for64Cu Radiolabeling
نویسندگان
چکیده
منابع مشابه
A new bifunctional chelator for copper radiopharmaceuticals: a cage amine ligand with a carboxylate functional group for conjugation to peptides.
A new sarcophagine cage amine ligand with a pendent carboxylate functional group has been synthesised; the ligand has been conjugated to tumour targeting peptides ([Tyr3]-octreotate and [Lys3]-bombesin) and the conjugates radiolabelled with copper-64.
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ژورنال
عنوان ژورنال: Molecular Pharmaceutics
سال: 2013
ISSN: 1543-8384,1543-8392
DOI: 10.1021/mp400686z